CN Patent
CN115141149A — 作为tyk2假激酶结构域抑制剂的杂环化合物及合成方法和用途
Assigned to Zhejiang Wenda Pharmaceutical Technology Co ltd · Expires 2022-10-04 · 4y expired
What this patent protects
本发明提供了作为TYK2假激酶(Pseudokinase,JH2)结构域抑制剂的杂环化合物及合成方法和用途。具体地,本发明提供了如式I所示的杂环化合物或其药学上可接受的盐,其中,各基团如文本中定义。本发明的杂环化合物具有优异的TYK2(JH2)选择抑制活性。
USPTO Abstract
本发明提供了作为TYK2假激酶(Pseudokinase,JH2)结构域抑制剂的杂环化合物及合成方法和用途。具体地,本发明提供了如式I所示的杂环化合物或其药学上可接受的盐,其中,各基团如文本中定义。本发明的杂环化合物具有优异的TYK2(JH2)选择抑制活性。
Drugs covered by this patent
- Sotyktu (DEUCRAVACITINIB) · Bristol-Myers Squibb
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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