CN Patent
CN114957381B — 新型氘代氰基类化合物、其制备方法、组合物及应用
Assigned to Guangzhou Anovent Pharmaceutical Co Ltd · Expires 2026-04-17 · 0y expired
What this patent protects
本发明公开了一种如式I所示的新型氘代氰基类化合物,或其药学上可接受的盐、异构体或前药。还公开了上述氘代化合物的制备方法、组合物及应用。该类化合物作为3CL蛋白酶抑制剂,在病毒抑制活性相当的基础上,实现了更优的药动学性质和治疗效果,成药性更好,式I如下所示:
USPTO Abstract
本发明公开了一种如式I所示的新型氘代氰基类化合物,或其药学上可接受的盐、异构体或前药。还公开了上述氘代化合物的制备方法、组合物及应用。该类化合物作为3CL蛋白酶抑制剂,在病毒抑制活性相当的基础上,实现了更优的药动学性质和治疗效果,成药性更好,式I如下所示:
Drugs covered by this patent
- Paxlovid (Copackaged) (Nirmatrelvir) · Pfizer
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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