CN Patent

CN114957236B — 一种2-酰基氨基噻唑类化合物的制备方法

Assigned to Nanjing Chia Tai Tianqing Pharmaceutical Co Ltd · Expires 2026-02-03 · 0y expired

What this patent protects

本发明涉及一种2-酰基氨基噻唑类化合物的制备方法,具体涉及一类阿伐曲泊帕中间体的制备方法,在该制备工艺中,使用四氢呋喃与DMSO的混合溶液做溶剂,使反应形成均相体系,进而使得该制备方法具有后处理简单、收率高和产品纯度高等优点,而且所采用的方法尤其适合工业化生产。

USPTO Abstract

本发明涉及一种2-酰基氨基噻唑类化合物的制备方法,具体涉及一类阿伐曲泊帕中间体的制备方法,在该制备工艺中,使用四氢呋喃与DMSO的混合溶液做溶剂,使反应形成均相体系,进而使得该制备方法具有后处理简单、收率高和产品纯度高等优点,而且所采用的方法尤其适合工业化生产。

Drugs covered by this patent

Patent Metadata

Patent number
CN114957236B
Jurisdiction
CN
Classification
Expires
2026-02-03
Drug substance claim
No
Drug product claim
No
Assignee
Nanjing Chia Tai Tianqing Pharmaceutical Co Ltd
Source
FDA Orange Book + USPTO grounding via Google Patents

Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.

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