CN Patent
CN114805216A — 奥拉帕利晶型及其制备方法
Assigned to Sichuan Kelun Pharmaceutical Research Institute Co Ltd · Expires 2022-07-29 · 4y expired
What this patent protects
本发明提供一种奥拉帕利晶型的制备方法,包括以下步骤:i)将奥拉帕利溶解在溶剂中得到奥拉帕利溶液;ii)将奥拉帕利溶液滴加到纯水或含水溶剂中;然后过滤干燥。采用本发明方法获得奥拉帕利晶型,因晶体尺寸较大,因此湿品中水含量低,解决了针状晶体常有的过滤困难、过滤洗涤效率差、烘干时间长、残留溶剂容易超标、杂质容易超标等技术问题。
USPTO Abstract
本发明提供一种奥拉帕利晶型的制备方法,包括以下步骤:i)将奥拉帕利溶解在溶剂中得到奥拉帕利溶液;ii)将奥拉帕利溶液滴加到纯水或含水溶剂中;然后过滤干燥。采用本发明方法获得奥拉帕利晶型,因晶体尺寸较大,因此湿品中水含量低,解决了针状晶体常有的过滤困难、过滤洗涤效率差、烘干时间长、残留溶剂容易超标、杂质容易超标等技术问题。
Drugs covered by this patent
- Lynparza (olaparib) · AstraZeneca
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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