CN Patent
CN114671889A — 一种取代三环吡啶酮衍生物的晶型及其制备方法
Assigned to Jiangsu Vcare Pharmatech Co Ltd · Expires 2022-06-28 · 4y expired
What this patent protects
本发明涉及一种取代三环吡啶酮衍生物的晶型及其制备方法,具体地涉及玛巴洛沙韦中间体7‑(苄氧基)‑3,4,12,12a‑四氢‑1H‑[1,4]噁嗪[3,4‑c]吡啶并[2,1‑f][1,2,4]三嗪‑6,8二酮的晶型,通过溶剂筛选得到晶型A,该晶型在高湿条件下稳定不易结块,且用该晶型为原料进行拆分得到的产物手性纯度高。
USPTO Abstract
本发明涉及一种取代三环吡啶酮衍生物的晶型及其制备方法,具体地涉及玛巴洛沙韦中间体7‑(苄氧基)‑3,4,12,12a‑四氢‑1H‑[1,4]噁嗪[3,4‑c]吡啶并[2,1‑f][1,2,4]三嗪‑6,8二酮的晶型,通过溶剂筛选得到晶型A,该晶型在高湿条件下稳定不易结块,且用该晶型为原料进行拆分得到的产物手性纯度高。
Drugs covered by this patent
- Xofluza (BALOXAVIR MARBOXIL) · Roche
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
Track this patent
Get a daily-checked alert when vulnerability score, expiry, classification, or assignee changes. Email, Slack, or Teams delivery. Pro: 50 watches, Free: 3.