CN Patent

CN114671889A — 一种取代三环吡啶酮衍生物的晶型及其制备方法

Assigned to Jiangsu Vcare Pharmatech Co Ltd · Expires 2022-06-28 · 4y expired

What this patent protects

本发明涉及一种取代三环吡啶酮衍生物的晶型及其制备方法,具体地涉及玛巴洛沙韦中间体7‑(苄氧基)‑3,4,12,12a‑四氢‑1H‑[1,4]噁嗪[3,4‑c]吡啶并[2,1‑f][1,2,4]三嗪‑6,8二酮的晶型,通过溶剂筛选得到晶型A,该晶型在高湿条件下稳定不易结块,且用该晶型为原料进行拆分得到的产物手性纯度高。

USPTO Abstract

本发明涉及一种取代三环吡啶酮衍生物的晶型及其制备方法,具体地涉及玛巴洛沙韦中间体7‑(苄氧基)‑3,4,12,12a‑四氢‑1H‑[1,4]噁嗪[3,4‑c]吡啶并[2,1‑f][1,2,4]三嗪‑6,8二酮的晶型,通过溶剂筛选得到晶型A,该晶型在高湿条件下稳定不易结块,且用该晶型为原料进行拆分得到的产物手性纯度高。

Drugs covered by this patent

Patent Metadata

Patent number
CN114671889A
Jurisdiction
CN
Classification
Expires
2022-06-28
Drug substance claim
No
Drug product claim
No
Assignee
Jiangsu Vcare Pharmatech Co Ltd
Source
FDA Orange Book + USPTO grounding via Google Patents

Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.

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