CN Patent
CN114502537A — 突变型idh2抑制剂及其应用
Assigned to Betta Pharmaceuticals Co Ltd · Expires 2022-05-13 · 4y expired
What this patent protects
一种作为突变型异柠檬酸脱氢酶2(IDH2)抑制剂的化合物(如式I所示)及其制备方法、药物组合物。还涉及上述化合物或其药物组合物在治疗突变型IDH2介导的疾病中的用途。IDH2抑制剂能够抑制携带最常见IDH2突变体的细胞中2‑HG的生成,是一种低毒性作用且高效靶向抗肿瘤药物的理想靶标。
USPTO Abstract
一种作为突变型异柠檬酸脱氢酶2(IDH2)抑制剂的化合物(如式I所示)及其制备方法、药物组合物。还涉及上述化合物或其药物组合物在治疗突变型IDH2介导的疾病中的用途。IDH2抑制剂能够抑制携带最常见IDH2突变体的细胞中2‑HG的生成,是一种低毒性作用且高效靶向抗肿瘤药物的理想靶标。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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