CN Patent
CN114478501A — 一种制备稳定的卡格列净半水合物晶型的方法
Assigned to Hangzhou Zhongmei Huadong Pharmaceutical Co Ltd · Expires 2022-05-13 · 4y expired
What this patent protects
本发明公开了一种稳定的卡格列净半水合物晶型及其制备方法,控制向卡格列净析晶体系中加入水的比例,以及在加入晶种之后快速搅拌,保温静置。该方法既能保证制得的卡格列净半水合物晶型纯度高,晶型又具备良好的形貌,能够不易发生转晶,保持良好的溶出性质。
USPTO Abstract
本发明公开了一种稳定的卡格列净半水合物晶型及其制备方法,控制向卡格列净析晶体系中加入水的比例,以及在加入晶种之后快速搅拌,保温静置。该方法既能保证制得的卡格列净半水合物晶型纯度高,晶型又具备良好的形貌,能够不易发生转晶,保持良好的溶出性质。
Drugs covered by this patent
- Invokana (CANAGLIFLOZIN) · Johnson & Johnson
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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