CN Patent
CN114437043B — 一种抗新冠药物Nirmatrelvir的制备方法
Assigned to Zhejiang Lepu Pharmaceutical Co ltd · Expires 2023-06-16 · 3y expired
What this patent protects
本发明公开了一种抗新冠药物Nirmatrelvir(化合物I)的制备方法。该制备方法以便宜易得的三氟乙酰‑L‑叔亮氨酸(化合物II)为起始原料,经过若干步反应即可得到Nirmatrelvir。本发明具有工艺简单可靠、综合成本低和易于商业化生产等优点。
USPTO Abstract
本发明公开了一种抗新冠药物Nirmatrelvir(化合物I)的制备方法。该制备方法以便宜易得的三氟乙酰‑L‑叔亮氨酸(化合物II)为起始原料,经过若干步反应即可得到Nirmatrelvir。本发明具有工艺简单可靠、综合成本低和易于商业化生产等优点。
Drugs covered by this patent
- Paxlovid (Copackaged) (Nirmatrelvir) · Pfizer
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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