CN114409653A — 一种桥环并嘧啶并环类化合物及其用途
Assigned to Suzhou Wentian Pharmaceutical Technology Co ltd · Expires 2022-04-29 · 4y expired
What this patent protects
本发明提供了一种桥环并嘧啶并环类化合物及其用途,桥环并嘧啶并环类化合物为下式(I)表示的化合物及其异构体或其药学上可接受的盐。本发明化合物能够应用于针对KRASG12C突变蛋白相关癌症的治疗药物中,KRASG12C突变蛋白相关癌症疾病选自:肺癌、结直肠癌、胰腺癌、胰腺癌、肝癌、胃癌、食道癌、胆管癌、乳腺癌、卵巢癌、子宫颈癌、黑色素瘤、脑胶质瘤、淋巴癌、白血病。
USPTO Abstract
本发明提供了一种桥环并嘧啶并环类化合物及其用途,桥环并嘧啶并环类化合物为下式(I)表示的化合物及其异构体或其药学上可接受的盐。本发明化合物能够应用于针对KRASG12C突变蛋白相关癌症的治疗药物中,KRASG12C突变蛋白相关癌症疾病选自:肺癌、结直肠癌、胰腺癌、胰腺癌、肝癌、胃癌、食道癌、胆管癌、乳腺癌、卵巢癌、子宫颈癌、黑色素瘤、脑胶质瘤、淋巴癌、白血病。
Drugs covered by this patent
- Krazati (ADAGRASIB) · Bristol-Myers Squibb
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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