CN Patent
CN114394957B — Met抑制剂盐酸特泊替尼的制备方法
Assigned to Wuhan Yujie Pharmaceutical Technology Co ltd · Expires 2023-05-09 · 3y expired
What this patent protects
本发明涉及一种MET抑制剂盐酸特泊替尼的制备方法。本发明采用市售易得的3‑甲基苄脒盐酸盐为起始物料,经环合反应,醚化反应,溴代反应及N‑烷基化反应合成目标产物。本发明所述的合成路线及制备方法,未见文献报道。本发明所述的方法有利于应用至大生产中。
USPTO Abstract
本发明涉及一种MET抑制剂盐酸特泊替尼的制备方法。本发明采用市售易得的3‑甲基苄脒盐酸盐为起始物料,经环合反应,醚化反应,溴代反应及N‑烷基化反应合成目标产物。本发明所述的合成路线及制备方法,未见文献报道。本发明所述的方法有利于应用至大生产中。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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