CN Patent
CN114366715A — 雷帕霉素自微乳注射剂及其制备方法及其应用
Assigned to Individual · Expires 2022-04-19 · 4y expired
What this patent protects
本发明提供了一种雷帕霉素自微乳注射剂,由药物母液和稀释剂组成;所述药物母液包括药物溶剂、抗氧剂和雷帕霉素;所述稀释剂包括表面活性剂和水。本发明雷帕霉素自微乳注射剂,由药物母液和稀释剂组成;把雷帕霉素溶解在药物溶剂中,稀释剂与母液混合稀释后,在表面活性剂的作用下,该液体就自组装形成微乳,同时,雷帕霉素被包封在微乳中,从而提高了雷帕霉素的溶解度,也提高了雷帕霉素稳定性。
USPTO Abstract
本发明提供了一种雷帕霉素自微乳注射剂,由药物母液和稀释剂组成;所述药物母液包括药物溶剂、抗氧剂和雷帕霉素;所述稀释剂包括表面活性剂和水。本发明雷帕霉素自微乳注射剂,由药物母液和稀释剂组成;把雷帕霉素溶解在药物溶剂中,稀释剂与母液混合稀释后,在表面活性剂的作用下,该液体就自组装形成微乳,同时,雷帕霉素被包封在微乳中,从而提高了雷帕霉素的溶解度,也提高了雷帕霉素稳定性。
Drugs covered by this patent
- Torisel (temsirolimus) · Pfizer
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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