CN114306261A — 巴洛沙韦酯片及其制备方法
Assigned to Aomei Pharmaceutical Hainan Co ltd · Expires 2022-04-12 · 4y expired
What this patent protects
本申请涉及于药物制剂技术领域,尤其涉及一种巴洛沙韦酯片及其制备方法,提供了一种巴洛沙韦酯片,其组成为巴洛沙韦酯、包合剂、填充剂、崩解剂、粘合剂、润滑剂及包衣剂;并且巴洛沙韦酯片采用环糊精包合技术,经过喷雾干燥制粒后,外加填充剂、崩解剂与润滑剂总混,最后压制成片剂。本发明制备的巴洛沙韦酯片溶出速率明显加快,提高了生物利用度,同时制备工艺稳定可控,产品质量稳定性好,用药安全性高,且便于服用、运输和储存,利于工业化生产。
USPTO Abstract
本申请涉及于药物制剂技术领域,尤其涉及一种巴洛沙韦酯片及其制备方法,提供了一种巴洛沙韦酯片,其组成为巴洛沙韦酯、包合剂、填充剂、崩解剂、粘合剂、润滑剂及包衣剂;并且巴洛沙韦酯片采用环糊精包合技术,经过喷雾干燥制粒后,外加填充剂、崩解剂与润滑剂总混,最后压制成片剂。本发明制备的巴洛沙韦酯片溶出速率明显加快,提高了生物利用度,同时制备工艺稳定可控,产品质量稳定性好,用药安全性高,且便于服用、运输和储存,利于工业化生产。
Drugs covered by this patent
- Xofluza (BALOXAVIR MARBOXIL) · Roche
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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