CN113662922A — 一种米拉贝隆缓释组合物及其制备方法和应用
Assigned to Chongqing Shisen Pharmaceutical Technology Co ltd · Expires 2021-11-19 · 4y expired
What this patent protects
本发明公开一种米拉贝隆缓释组合物及其制备方法和应用。所述组合物包含:活性成分米拉贝隆和药用辅料;所述药用辅料至少含有抗氧化剂,所述抗氧化剂选自二丁基羟基甲苯、丁基羟基茴香醚和维生素E中的至少一种。在氮气保护下制备含有米拉贝隆和胶凝剂、凝胶增强剂和抗氧化剂的共熔体混合物,将共熔体混合物用水冷粉碎机进行粉碎,形成活性成分米拉贝隆分布均匀的颗粒。制备得到的缓释片具有优异的缓释效果。
USPTO Abstract
本发明公开一种米拉贝隆缓释组合物及其制备方法和应用。所述组合物包含:活性成分米拉贝隆和药用辅料;所述药用辅料至少含有抗氧化剂,所述抗氧化剂选自二丁基羟基甲苯、丁基羟基茴香醚和维生素E中的至少一种。在氮气保护下制备含有米拉贝隆和胶凝剂、凝胶增强剂和抗氧化剂的共熔体混合物,将共熔体混合物用水冷粉碎机进行粉碎,形成活性成分米拉贝隆分布均匀的颗粒。制备得到的缓释片具有优异的缓释效果。
Drugs covered by this patent
- Myrbetriq (MIRABEGRON) · Apgdi
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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