CN Patent

CN113603708B — 一种具有大环骨架结构的cdk9抑制剂的制备及其应用

Assigned to China Pharmaceutical University · Expires 2023-08-11 · 3y expired

What this patent protects

本发明公开了一种具有大环骨架结构的CDK9抑制剂的制备及其应用,该类化合物可以有效地抑制CDK9蛋白的活性并具有较好的CDK9选择性;本发明还公开了上述化合物的制备方法及其在预防和/或治疗肿瘤相关疾病中的应用,包括神经胶质瘤、各类白血病、淋巴癌、肝癌、胃癌、前列腺癌、卵巢癌、乳腺癌、肺癌等。

USPTO Abstract

本发明公开了一种具有大环骨架结构的CDK9抑制剂的制备及其应用,该类化合物可以有效地抑制CDK9蛋白的活性并具有较好的CDK9选择性;本发明还公开了上述化合物的制备方法及其在预防和/或治疗肿瘤相关疾病中的应用,包括神经胶质瘤、各类白血病、淋巴癌、肝癌、胃癌、前列腺癌、卵巢癌、乳腺癌、肺癌等。

Drugs covered by this patent

Patent Metadata

Patent number
CN113603708B
Jurisdiction
CN
Classification
Expires
2023-08-11
Drug substance claim
No
Drug product claim
No
Assignee
China Pharmaceutical University
Source
FDA Orange Book + USPTO grounding via Google Patents

Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.

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