CN113248500B — 氮杂吲哚嘧啶胺杂环化合物及其制备方法和应用
Assigned to China Pharmaceutical University · Expires 2021-10-19 · 5y expired
What this patent protects
本发明公开了一种氮杂吲哚嘧啶胺杂环化合物及其制备方法和应用,所述化合物如式(S)所示。本发明的化合物能抑制癌症的恶性增殖,治疗效果好、毒性低,具有良好药物代谢特性、不易产生耐药性,可用于制备治疗癌症或肿瘤相关疾病药物,所述癌症或肿瘤相关疾病包括多发性骨髓瘤、白血病、乳腺癌、前列腺癌、肺癌、肝癌、胃癌、骨癌、脑癌、头颈癌、肠癌、胰腺癌、膀胱癌、睾丸癌、卵巢癌以及子宫内膜癌。
USPTO Abstract
本发明公开了一种氮杂吲哚嘧啶胺杂环化合物及其制备方法和应用,所述化合物如式(S)所示。本发明的化合物能抑制癌症的恶性增殖,治疗效果好、毒性低,具有良好药物代谢特性、不易产生耐药性,可用于制备治疗癌症或肿瘤相关疾病药物,所述癌症或肿瘤相关疾病包括多发性骨髓瘤、白血病、乳腺癌、前列腺癌、肺癌、肝癌、胃癌、骨癌、脑癌、头颈癌、肠癌、胰腺癌、膀胱癌、睾丸癌、卵巢癌以及子宫内膜癌。
Drugs covered by this patent
- Verzenio (abemaciclib) · Eli Lilly
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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