CN Patent
CN113214261A — 一种依鲁替尼晶型a的纯化方法
Assigned to SYNCOZYMES (SHANGHAI) CO Ltd · Expires 2021-08-06 · 5y expired
What this patent protects
本发明公开了一种依鲁替尼晶型A的纯化方法,该方法为利用晶型转化实现依鲁替尼晶型A的纯化,具体过程为将依鲁替尼晶型A粗品溶解、加入晶种E后得到依鲁替尼晶型E,再将晶型E溶解、结晶得到纯度更高的依鲁替尼晶型A。本发明所述的依鲁替尼晶型A的纯化方法工艺简单、产率高,解决了依鲁替尼结晶A中难除杂质的纯化问题。
USPTO Abstract
本发明公开了一种依鲁替尼晶型A的纯化方法,该方法为利用晶型转化实现依鲁替尼晶型A的纯化,具体过程为将依鲁替尼晶型A粗品溶解、加入晶种E后得到依鲁替尼晶型E,再将晶型E溶解、结晶得到纯度更高的依鲁替尼晶型A。本发明所述的依鲁替尼晶型A的纯化方法工艺简单、产率高,解决了依鲁替尼结晶A中难除杂质的纯化问题。
Drugs covered by this patent
- Imbruvica (ibrutinib) · AbbVie
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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