CN Patent
CN113045565A — 新型K-Ras G12C抑制剂
Assigned to Wigen Biomedicine Technology Shanghai Co Ltd · Expires 2021-06-29 · 5y expired
What this patent protects
本发明涉及一类式(1)所示的化合物及其制备方法,及式(1)化合物及其各光学异构体、各晶型、药学上可接受的盐作为G12C突变体K‑Ras蛋白不可逆抑制剂在抗肿瘤等Ras相关疾病的药物制备中的用途。
USPTO Abstract
本发明涉及一类式(1)所示的化合物及其制备方法,及式(1)化合物及其各光学异构体、各晶型、药学上可接受的盐作为G12C突变体K‑Ras蛋白不可逆抑制剂在抗肿瘤等Ras相关疾病的药物制备中的用途。
Drugs covered by this patent
- Krazati (ADAGRASIB) · Bristol-Myers Squibb
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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