CN Patent
CN113004269B — Kras-G12C抑制剂杂环化合物
Assigned to Capital Pharmaceutical Holdings Beijing Co ltd · Expires 2024-11-05 · 2y expired
What this patent protects
本申请涉及一类式I所示Kras‑G12C抑制剂杂环化合物,及其制备方法和该类化合物在肿瘤疾病,如肺癌、结直肠癌和胰腺癌等中的预防和治疗用途。在制备过程中,通过SN2反应、上保护、偶联反应、脱保户、缩合反应等一系列反应,得到通式化合物I。
USPTO Abstract
本申请涉及一类式I所示Kras‑G12C抑制剂杂环化合物,及其制备方法和该类化合物在肿瘤疾病,如肺癌、结直肠癌和胰腺癌等中的预防和治疗用途。在制备过程中,通过SN2反应、上保护、偶联反应、脱保户、缩合反应等一系列反应,得到通式化合物I。
Drugs covered by this patent
- Krazati (ADAGRASIB) · Bristol-Myers Squibb
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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