CN Patent

CN113004269B — Kras-G12C抑制剂杂环化合物

Assigned to Capital Pharmaceutical Holdings Beijing Co ltd · Expires 2024-11-05 · 2y expired

What this patent protects

本申请涉及一类式I所示Kras‑G12C抑制剂杂环化合物,及其制备方法和该类化合物在肿瘤疾病,如肺癌、结直肠癌和胰腺癌等中的预防和治疗用途。在制备过程中,通过SN2反应、上保护、偶联反应、脱保户、缩合反应等一系列反应,得到通式化合物I。

USPTO Abstract

本申请涉及一类式I所示Kras‑G12C抑制剂杂环化合物,及其制备方法和该类化合物在肿瘤疾病,如肺癌、结直肠癌和胰腺癌等中的预防和治疗用途。在制备过程中,通过SN2反应、上保护、偶联反应、脱保户、缩合反应等一系列反应,得到通式化合物I。

Drugs covered by this patent

Patent Metadata

Patent number
CN113004269B
Jurisdiction
CN
Classification
Expires
2024-11-05
Drug substance claim
No
Drug product claim
No
Assignee
Capital Pharmaceutical Holdings Beijing Co ltd
Source
FDA Orange Book + USPTO grounding via Google Patents

Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.

Track this patent

Get a daily-checked alert when vulnerability score, expiry, classification, or assignee changes. Email, Slack, or Teams delivery. Pro: 50 watches, Free: 3.