CN Patent
CN112888691B — 吡咯并[2,3-d]嘧啶甲苯磺酸盐、其结晶形式以及有关的制备方法和中间体
Assigned to Pfizer Inc · Expires 2023-10-31 · 3y expired
What this patent protects
本发明公开了1‑((2S,5R)‑5‑((7H‑吡咯并[2,3‑d]嘧啶‑4‑基)氨基)‑2‑甲基哌啶‑1‑基)丙‑2‑烯‑1‑酮的新的对甲苯磺酸盐和所述盐的结晶多晶型形式1,含有它们的药物组合物,以及其制备及用途。本发明也公开了1‑((2S,5R)‑5‑((7H‑吡咯并[2,3‑d]嘧啶‑4‑基)氨基)‑2‑甲基哌啶‑1‑基)丙‑2‑烯‑1‑酮的新的磷酸盐,含有它们的药物组合物,以及其制备及用途。
USPTO Abstract
本发明公开了1‑((2S,5R)‑5‑((7H‑吡咯并[2,3‑d]嘧啶‑4‑基)氨基)‑2‑甲基哌啶‑1‑基)丙‑2‑烯‑1‑酮的新的对甲苯磺酸盐和所述盐的结晶多晶型形式1,含有它们的药物组合物,以及其制备及用途。本发明也公开了1‑((2S,5R)‑5‑((7H‑吡咯并[2,3‑d]嘧啶‑4‑基)氨基)‑2‑甲基哌啶‑1‑基)丙‑2‑烯‑1‑酮的新的磷酸盐,含有它们的药物组合物,以及其制备及用途。
Drugs covered by this patent
- Litfulo (Ritlecitinib Tosylate) · Pfizer
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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