CN Patent
CN112824410A — 氮杂七元环类抑制剂及其制备方法和应用
Assigned to Shanghai Zejing Pharmaceutical Technology Co ltd · Expires 2021-05-21 · 5y expired
What this patent protects
本发明涉及氮杂七元环类抑制剂及其制备方法和应用。具体地,本发明化合物具有式(I)所示结构,本发明还公开了所述化合物的制备方法及其作为KRAS G12C 抑制剂的用途,对KRAS G12C 具有很好的选择性抑制作用且具有更好的药效学、药代动力学性能和更低的毒副作用。
USPTO Abstract
本发明涉及氮杂七元环类抑制剂及其制备方法和应用。具体地,本发明化合物具有式(I)所示结构,本发明还公开了所述化合物的制备方法及其作为KRAS G12C 抑制剂的用途,对KRAS G12C 具有很好的选择性抑制作用且具有更好的药效学、药代动力学性能和更低的毒副作用。
Drugs covered by this patent
- Krazati (ADAGRASIB) · Bristol-Myers Squibb
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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