CN Patent
CN112812052B — 一种治疗溃疡性结肠炎的化合物及其制备方法和用途
Assigned to Chengdu Achi Biopharmaceutical Technology Co ltd · Expires 2023-12-01 · 2y expired
What this patent protects
本发明提供了一种治疗溃疡性结肠炎的化合物,具有式I所示结构。本发明提供的化合物能够显著抑制患结肠炎时结肠组织中TNF‑α、IL‑1β和IL‑6等促炎因子的异常分泌,抑制炎性细胞浸润,维持肠上皮和隐窝腺的完整,能够有效减轻炎症,改善结肠缩短和肠壁增厚症状,在制备治疗溃疡性结肠炎的药物中具有优异的潜在应用价值,为临床提供了新的选择。
USPTO Abstract
本发明提供了一种治疗溃疡性结肠炎的化合物,具有式I所示结构。本发明提供的化合物能够显著抑制患结肠炎时结肠组织中TNF‑α、IL‑1β和IL‑6等促炎因子的异常分泌,抑制炎性细胞浸润,维持肠上皮和隐窝腺的完整,能够有效减轻炎症,改善结肠缩短和肠壁增厚症状,在制备治疗溃疡性结肠炎的药物中具有优异的潜在应用价值,为临床提供了新的选择。
Drugs covered by this patent
- Velsipity (Etrasimod Arginine) · Pfizer Inc.
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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