CN Patent
CN112679438A — 制备司美替尼的方法
Assigned to Wuhan Jiuzhou Yumin Medical Technology Co ltd · Expires 2021-04-20 · 5y expired
What this patent protects
本发明涉及一种制备MEK1/2抑制剂司美替尼的方法,本发明的合成路线经三步反应合成得到司美替尼,其合成方法的后处理均无需柱层析分离,反应产物直接析出干燥即可。利用本发明所述的合成制备方法,其能够快速、有效地制备获得司美替尼。
USPTO Abstract
本发明涉及一种制备MEK1/2抑制剂司美替尼的方法,本发明的合成路线经三步反应合成得到司美替尼,其合成方法的后处理均无需柱层析分离,反应产物直接析出干燥即可。利用本发明所述的合成制备方法,其能够快速、有效地制备获得司美替尼。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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