CN Patent
CN112574200B — Btk和/或btk的突变体c481s的小分子抑制剂
Assigned to Anrun Pharmaceutical Technology Suzhou Co ltd · Expires 2021-06-11 · 5y expired
What this patent protects
本发明涉及一种BTK和/或BTK的突变体C481S的小分子抑制剂,其包括式I所示的化合物或其烯醇化物、立体异构体、互变异构体、水合物、溶剂化物或药学上可接受的盐,上述化合物可用于制备预防和/或治疗BTK的活性异常和/或BTK的突变体C481S的活性异常有关的疾病的药物,如自身免疫性疾病、炎症性疾病或癌症。
USPTO Abstract
本发明涉及一种BTK和/或BTK的突变体C481S的小分子抑制剂,其包括式I所示的化合物或其烯醇化物、立体异构体、互变异构体、水合物、溶剂化物或药学上可接受的盐,上述化合物可用于制备预防和/或治疗BTK的活性异常和/或BTK的突变体C481S的活性异常有关的疾病的药物,如自身免疫性疾病、炎症性疾病或癌症。
Drugs covered by this patent
- Zelboraf (vemurafenib) · Hoffmann La Roche
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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