CN Patent
CN112500358B — 赛乐西帕晶型及其制备方法
Assigned to Jiangsu Hansoh Pharmaceutical Group Co Ltd · Expires 2022-03-15 · 4y expired
What this patent protects
本发明涉及具有改善性质的赛乐西帕新晶型及其制备方法,该方法采用循环析晶的方式得到一种赛乐西帕晶型A。与传统赛乐西帕晶型相比,该赛乐西帕晶型A的熔点高,稳定性好,晶型纯度高,有关物质含量低,工艺条件温和,适合大规模生产,包含该晶型的药物组合物及剂型可用于治疗肺动脉高压疾病。
USPTO Abstract
本发明涉及具有改善性质的赛乐西帕新晶型及其制备方法,该方法采用循环析晶的方式得到一种赛乐西帕晶型A。与传统赛乐西帕晶型相比,该赛乐西帕晶型A的熔点高,稳定性好,晶型纯度高,有关物质含量低,工艺条件温和,适合大规模生产,包含该晶型的药物组合物及剂型可用于治疗肺动脉高压疾病。
Drugs covered by this patent
- Uptravi (SELEXIPAG) · AstraZeneca
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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