CN Patent
CN112300081A — 噁拉戈利的中间体及其制备方法和应用
Assigned to Shanghai Dude Pharmaceutical Technology Co ltd · Expires 2021-02-02 · 5y expired
What this patent protects
本发明提供了一种新的噁拉戈利重要中间体化合物1制备方法,同时还提供了两个新的中间体化合物5和6。由新的中间体化合物5开始,使得现有技术的的五步合成缩减为三步,不仅收率大大提高,而且反应能耗低、“三废”少、制备周期短,更易于工业化放大生产。
USPTO Abstract
本发明提供了一种新的噁拉戈利重要中间体化合物1制备方法,同时还提供了两个新的中间体化合物5和6。由新的中间体化合物5开始,使得现有技术的的五步合成缩减为三步,不仅收率大大提高,而且反应能耗低、“三废”少、制备周期短,更易于工业化放大生产。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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