CN Patent
CN112142662B — 一种甲磺酸乐伐替尼的制备方法
Assigned to Nanjing Finetech Chemical Co ltd · Expires 2022-03-08 · 4y expired
What this patent protects
本发明涉及一种甲磺酸乐伐替尼的制备方法,具体涉及以4‑氯‑6‑氰基‑7‑甲氧基喹啉和2‑氯‑4‑羟基苯胺甲酸环丙酰胺为原料,经取代反应、水解反应两步高效合成甲磺酸乐伐替尼,本发明提供的甲磺酸乐伐替尼的制备方法是一种步骤短、高收率、低成本、三废少、产品纯度好、适宜工业化的制备方法。
USPTO Abstract
本发明涉及一种甲磺酸乐伐替尼的制备方法,具体涉及以4‑氯‑6‑氰基‑7‑甲氧基喹啉和2‑氯‑4‑羟基苯胺甲酸环丙酰胺为原料,经取代反应、水解反应两步高效合成甲磺酸乐伐替尼,本发明提供的甲磺酸乐伐替尼的制备方法是一种步骤短、高收率、低成本、三废少、产品纯度好、适宜工业化的制备方法。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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