CN112137981A — 富马酸丙酚替诺福韦片及其制备工艺
Assigned to Chengdu Jingfu Pharmaceutical Technology Co ltd · Expires 2020-12-29 · 5y expired
What this patent protects
本发明公开了富马酸丙酚替诺福韦片及其制备工艺,富马酸丙酚替诺福韦片将以下配方制成1000片富马酸丙酚替诺福韦片,所述配方包括内加配方、外加配方和包衣预混剂:内加配方由以下组分组成:富马酸丙酚替诺福韦25g、乳糖95g、微晶纤维素50g、交联羧甲纤维素钠10g、硬脂酸镁1g、碳酸氢钠0.5g和依地酸二钠0.5g;外加配方由以下组分组成:微晶纤维素10g、交联羧甲纤维素钠4g、硬脂酸镁2g和碳酸氢钠1g;包衣预混剂8g。本发明通过同时对内加配方和外加配方进行改进,从内到外双重稳定作用,提高了富马酸丙酚替诺福韦片的稳定性。
USPTO Abstract
本发明公开了富马酸丙酚替诺福韦片及其制备工艺,富马酸丙酚替诺福韦片将以下配方制成1000片富马酸丙酚替诺福韦片,所述配方包括内加配方、外加配方和包衣预混剂:内加配方由以下组分组成:富马酸丙酚替诺福韦25g、乳糖95g、微晶纤维素50g、交联羧甲纤维素钠10g、硬脂酸镁1g、碳酸氢钠0.5g和依地酸二钠0.5g;外加配方由以下组分组成:微晶纤维素10g、交联羧甲纤维素钠4g、硬脂酸镁2g和碳酸氢钠1g;包衣预混剂8g。本发明通过同时对内加配方和外加配方进行改进,从内到外双重稳定作用,提高了富马酸丙酚替诺福韦片的稳定性。
Drugs covered by this patent
- Emtriva (EMTRICITABINE) · Gilead Sciences
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
Track this patent
Get a daily-checked alert when vulnerability score, expiry, classification, or assignee changes. Email, Slack, or Teams delivery. Pro: 50 watches, Free: 3.