CN Patent

CN111825678A — 一种卡马替尼的制备方法

Assigned to Individual · Expires 2020-10-27 · 6y expired

What this patent protects

本发明提供了一种卡马替尼的制备方法,发明人经过广泛而深入的研究,通过大量筛选和测试,利用式Ⅲ化合物为原料,经过水解反应、甲基化反应,得到式Ⅰ化合物即卡马替尼。该方法反应条件温和、环境友好、能耗低,所得产物纯度好且收率高,适宜工业化大生产。

USPTO Abstract

本发明提供了一种卡马替尼的制备方法,发明人经过广泛而深入的研究,通过大量筛选和测试,利用式Ⅲ化合物为原料,经过水解反应、甲基化反应,得到式Ⅰ化合物即卡马替尼。该方法反应条件温和、环境友好、能耗低,所得产物纯度好且收率高,适宜工业化大生产。

Drugs covered by this patent

Patent Metadata

Patent number
CN111825678A
Jurisdiction
CN
Classification
Expires
2020-10-27
Drug substance claim
No
Drug product claim
No
Assignee
Individual
Source
FDA Orange Book + USPTO grounding via Google Patents

Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.

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