CN Patent

CN111620873B — 一类含哌啶的吡咯并[2,3-d]嘧啶衍生物及其制备和用途

Assigned to Shenyang Pharmaceutical University · Expires 2021-12-28 · 4y expired

What this patent protects

本发明涉及通式I或通式II所示的含哌啶的吡咯并[2,3‑d]嘧啶衍生物及使用和制备方法。本发明还涉及通式I或II的化合物具有强的JAK激酶的抑制作用,并且还涉及该类化合物在制备用于治疗和/或预防由于JAK异常表达所引起疾病的药物中的应用,特别是在制备治疗炎症/自身免疫疾病、纤维化和癌症的药物中的用途。

USPTO Abstract

本发明涉及通式I或通式II所示的含哌啶的吡咯并[2,3‑d]嘧啶衍生物及使用和制备方法。本发明还涉及通式I或II的化合物具有强的JAK激酶的抑制作用,并且还涉及该类化合物在制备用于治疗和/或预防由于JAK异常表达所引起疾病的药物中的应用,特别是在制备治疗炎症/自身免疫疾病、纤维化和癌症的药物中的用途。

Drugs covered by this patent

Patent Metadata

Patent number
CN111620873B
Jurisdiction
CN
Classification
Expires
2021-12-28
Drug substance claim
No
Drug product claim
No
Assignee
Shenyang Pharmaceutical University
Source
FDA Orange Book + USPTO grounding via Google Patents

Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.

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