CN Patent
CN111620863A — 阿曲波帕的制备方法
Assigned to Suzhou Miracpharma Technology Co Ltd · Expires 2020-09-04 · 6y expired
What this patent protects
本发明揭示了一种阿曲波帕(Avatrombopag)的制备方法,以6‑氨基‑5‑氯‑3‑吡啶苯甲酸为起始原料,依次进行环化、酰胺化和水解等反应,制得目标产物阿曲波帕。该制备过程原料易得、快捷方便、经济环保,尤其克服了现行工艺原料中双氯选择性差等问题,适于大规模工业化生产。
USPTO Abstract
本发明揭示了一种阿曲波帕(Avatrombopag)的制备方法,以6‑氨基‑5‑氯‑3‑吡啶苯甲酸为起始原料,依次进行环化、酰胺化和水解等反应,制得目标产物阿曲波帕。该制备过程原料易得、快捷方便、经济环保,尤其克服了现行工艺原料中双氯选择性差等问题,适于大规模工业化生产。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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