CN Patent
CN111440151A — 制备抗肿瘤药普拉赛替尼的方法
Assigned to Individual · Expires 2020-07-24 · 6y expired
What this patent protects
本发明涉及一种制备抗肿瘤药普拉塞替尼的方法。本发明经卤代、脱甲基保护基、酰胺缩合反应三步能够快速、有效地制备获得普拉塞替尼,本发明所述的制备方法,其路线反应步数少,大幅度减少了反应步数,提高了反应的总收率,有效降低了终产物成本。
USPTO Abstract
本发明涉及一种制备抗肿瘤药普拉塞替尼的方法。本发明经卤代、脱甲基保护基、酰胺缩合反应三步能够快速、有效地制备获得普拉塞替尼,本发明所述的制备方法,其路线反应步数少,大幅度减少了反应步数,提高了反应的总收率,有效降低了终产物成本。
Drugs covered by this patent
- Gavreto (PRALSETINIB) · Rigel Pharms
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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