CN Patent
CN111377944A — Baloxavir marboxil晶型及其制备方法
Assigned to Sunshine Lake Pharma Co Ltd · Expires 2020-07-07 · 6y expired
What this patent protects
本发明提供了一种Baloxavir marboxil晶型A和晶型B及其制备方法,属于药物化学领域。所述晶型具有良好的溶解度、稳定性等其他性质。本发明所述制备方法通过将Baloxavir marboxil固体与有机溶剂混合,然后加入反溶剂或者不加反溶剂,搅拌,过滤,可得Baloxavir marboxil晶型A和晶型B;所述制备方法操作简单,条件温和。
USPTO Abstract
本发明提供了一种Baloxavir marboxil晶型A和晶型B及其制备方法,属于药物化学领域。所述晶型具有良好的溶解度、稳定性等其他性质。本发明所述制备方法通过将Baloxavir marboxil固体与有机溶剂混合,然后加入反溶剂或者不加反溶剂,搅拌,过滤,可得Baloxavir marboxil晶型A和晶型B;所述制备方法操作简单,条件温和。
Drugs covered by this patent
- Xofluza (BALOXAVIR MARBOXIL) · Roche
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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