CN Patent

CN111217792B — 一种来那度胺b晶型的制备方法

Assigned to Cinkate Pharm Tech (shanghai) Co ltd · Expires 2021-09-28 · 5y expired

What this patent protects

本发明提供一种来那度胺B晶型的制备方法。具体地,本发明提供的方法包括步骤:(1)使原料来那度胺溶解于醇中,得到含来那度胺的溶液;和(2)向步骤(1)得到的含来那度胺的溶液中加入水,析晶得到来那度胺B晶型;其中,所述的醇选自下组:1,3‑丙二醇、1,2‑丙二醇,或其组合。本发明方法具有高稳定性和可靠性。

USPTO Abstract

本发明提供一种来那度胺B晶型的制备方法。具体地,本发明提供的方法包括步骤:(1)使原料来那度胺溶解于醇中,得到含来那度胺的溶液;和(2)向步骤(1)得到的含来那度胺的溶液中加入水,析晶得到来那度胺B晶型;其中,所述的醇选自下组:1,3‑丙二醇、1,2‑丙二醇,或其组合。本发明方法具有高稳定性和可靠性。

Drugs covered by this patent

Patent Metadata

Patent number
CN111217792B
Jurisdiction
CN
Classification
Expires
2021-09-28
Drug substance claim
No
Drug product claim
No
Assignee
Cinkate Pharm Tech (shanghai) Co ltd
Source
FDA Orange Book + USPTO grounding via Google Patents

Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.

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