CN Patent
CN111138436A — 伊布替尼晶型a单晶及其制备方法
Assigned to Lunan Pharmaceutical Group Corp · Expires 2020-05-12 · 6y expired
What this patent protects
本发明属于化学药物制备技术领域,具体公开了伊布替尼晶型A单晶及其制备方法,将伊布替尼晶型A溶于良溶剂中,完全溶解后加入不良溶剂过滤析晶即得。经过本发明的技术方案可以培养出更多形状良好的伊布替尼晶型A单晶,工艺简单,单晶培养时间短,晶型稳定,易于挑选,在室温下挑选不易融化。
USPTO Abstract
本发明属于化学药物制备技术领域,具体公开了伊布替尼晶型A单晶及其制备方法,将伊布替尼晶型A溶于良溶剂中,完全溶解后加入不良溶剂过滤析晶即得。经过本发明的技术方案可以培养出更多形状良好的伊布替尼晶型A单晶,工艺简单,单晶培养时间短,晶型稳定,易于挑选,在室温下挑选不易融化。
Drugs covered by this patent
- Imbruvica (ibrutinib) · AbbVie
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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