CN Patent

CN111004257B — 制备RET抑制剂Selpercatinib的方法

Assigned to Wuhan Jiuzhou Yumin Medical Technology Co ltd · Expires 2021-06-29 · 5y expired

What this patent protects

本发明涉及一种制备RET抑制剂Selpercatinib的方法。本发明所述的制备方法,其卤化反应条件更温和,反应操作步骤及后处理更简便,反应步骤少,大幅度提高了反应的总产率,产物纯度达到99.0%以上。

USPTO Abstract

本发明涉及一种制备RET抑制剂Selpercatinib的方法。本发明所述的制备方法,其卤化反应条件更温和,反应操作步骤及后处理更简便,反应步骤少,大幅度提高了反应的总产率,产物纯度达到99.0%以上。

Drugs covered by this patent

Patent Metadata

Patent number
CN111004257B
Jurisdiction
CN
Classification
Expires
2021-06-29
Drug substance claim
No
Drug product claim
No
Assignee
Wuhan Jiuzhou Yumin Medical Technology Co ltd
Source
FDA Orange Book + USPTO grounding via Google Patents

Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.

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