CN Patent

CN110724137B — 一种噻吩类衍生物及其制备方法与应用

Assigned to Guangdong University of Technology · Expires 2021-03-30 · 5y expired

What this patent protects

本发明涉及药物化学技术领域,尤其涉及一种噻吩类衍生物及其制备方法与应用。本发明公开了一种具有式(Ⅰ)结构的噻吩类衍生物或其药学上可接受的盐、所述药学上可接受的盐的溶剂化合物、对映异构体、非对映异构体、互变异构体、消旋体或其组合。该化合物具有较好的水溶性、对酪氨酸激酶和肿瘤细胞有较强的抑制作用。

USPTO Abstract

本发明涉及药物化学技术领域,尤其涉及一种噻吩类衍生物及其制备方法与应用。本发明公开了一种具有式(Ⅰ)结构的噻吩类衍生物或其药学上可接受的盐、所述药学上可接受的盐的溶剂化合物、对映异构体、非对映异构体、互变异构体、消旋体或其组合。该化合物具有较好的水溶性、对酪氨酸激酶和肿瘤细胞有较强的抑制作用。

Drugs covered by this patent

Patent Metadata

Patent number
CN110724137B
Jurisdiction
CN
Classification
Expires
2021-03-30
Drug substance claim
No
Drug product claim
No
Assignee
Guangdong University of Technology
Source
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Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.

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