CN Patent
CN110650963B — Gdc-0077的多晶型物和固体形式及其制备方法
Assigned to F Hoffmann La Roche AG · Expires 2022-09-27 · 4y expired
What this patent protects
本发明涉及具有以下式I结构的(5)‑2‑((2‑((5)‑4‑(二氟甲基)‑2‑氧代噁唑烷‑3‑基)‑5,6‑二氢苯并[f]咪唑并[1,2‑J][1,4]氧氮杂 ‑9‑基)氨基)丙酰胺(GDC‑0077)(或其立体异构体、几何异构体、互变异构体及药用盐)的结晶多晶型物形式,及制备所述多晶型物形式的方法,
USPTO Abstract
本发明涉及具有以下式I结构的(5)‑2‑((2‑((5)‑4‑(二氟甲基)‑2‑氧代噁唑烷‑3‑基)‑5,6‑二氢苯并[f]咪唑并[1,2‑J][1,4]氧氮杂 ‑9‑基)氨基)丙酰胺(GDC‑0077)(或其立体异构体、几何异构体、互变异构体及药用盐)的结晶多晶型物形式,及制备所述多晶型物形式的方法,
Drugs covered by this patent
- Itovebi (INAVOLISIB) · Genentech Inc
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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