CN Patent
CN110563733A — 作为选择性btk抑制剂的咪唑并吡嗪类化合物
Assigned to An Dikang (wuxi) Biotechnology Co Ltd · Expires 2019-12-13 · 6y expired
What this patent protects
本发明涉及作为选择性布鲁顿酪氨酸激酶(BTK)抑制剂的咪唑并吡嗪类化合物。具体而言,本发明公开了(S)‑4‑(8‑氨基‑3‑(1‑(丁‑2‑炔酰基)吡咯烷‑2‑基)咪唑并[1,5‑a]吡嗪‑1‑基)‑N‑(吡啶‑2‑基)苯甲酰胺和其光学异构体的氘代化合物,或药学上可接受的盐或涉及含有这类化合物的药物组合物,以及他们在治疗BTK介导的疾病中的用途。
USPTO Abstract
本发明涉及作为选择性布鲁顿酪氨酸激酶(BTK)抑制剂的咪唑并吡嗪类化合物。具体而言,本发明公开了(S)‑4‑(8‑氨基‑3‑(1‑(丁‑2‑炔酰基)吡咯烷‑2‑基)咪唑并[1,5‑a]吡嗪‑1‑基)‑N‑(吡啶‑2‑基)苯甲酰胺和其光学异构体的氘代化合物,或药学上可接受的盐或涉及含有这类化合物的药物组合物,以及他们在治疗BTK介导的疾病中的用途。
Drugs covered by this patent
- Calquence (ACALABRUTINIB) · AstraZeneca
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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