CN Patent
CN110407819B — 一种作为预防外科手术并发症的凝血酶受体拮抗剂
Assigned to Mudanjiang Medical University · Expires 2020-06-26 · 6y expired
What this patent protects
提供一种沃拉帕沙衍生物及其制备方法,所述化合物的结构如式I所示,其中R 1 选自氢、卤素、C1‑5烷基、氟代C1‑5烷基;所述化合物具有优异的PAR‑1抑制活性,尤其适用外科手术中预防并发症的出现,也有望替代沃拉帕沙成为一种有潜力的治疗心肌梗死、冠状动脉疾病的新药。
USPTO Abstract
提供一种沃拉帕沙衍生物及其制备方法,所述化合物的结构如式I所示,其中R 1 选自氢、卤素、C1‑5烷基、氟代C1‑5烷基;所述化合物具有优异的PAR‑1抑制活性,尤其适用外科手术中预防并发症的出现,也有望替代沃拉帕沙成为一种有潜力的治疗心肌梗死、冠状动脉疾病的新药。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
Track this patent
Get a daily-checked alert when vulnerability score, expiry, classification, or assignee changes. Email, Slack, or Teams delivery. Pro: 50 watches, Free: 3.