CN Patent
CN110272419A — 二氢吡啶并酞嗪酮衍生物、其制备方法及应用
Assigned to Shanghai Allist Pharmaceuticals Inc · Expires 2019-09-24 · 7y expired
What this patent protects
本发明涉及下述通式(I)所示的二氢吡啶并酞嗪酮衍生物、其制备方法与应用,式中R 1 、R 2 、R 3 、m、n、环A和环B如说明书中所定义。本发明所述二氢吡啶并酞嗪酮衍生物具有良好的PARP抑制活性,可用于治疗或预防因抑制PARP活性而改善的疾病。
USPTO Abstract
本发明涉及下述通式(I)所示的二氢吡啶并酞嗪酮衍生物、其制备方法与应用,式中R 1 、R 2 、R 3 、m、n、环A和环B如说明书中所定义。本发明所述二氢吡啶并酞嗪酮衍生物具有良好的PARP抑制活性,可用于治疗或预防因抑制PARP活性而改善的疾病。
Drugs covered by this patent
- Talzenna (Talazoparib Tosylate) · Pfizer Inc.
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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