CN Patent
CN110114361B — Nrf2化合物
Assigned to GlaxoSmithKline Intellectual Property Development Ltd · Expires 2022-04-12 · 4y expired
What this patent protects
本发明涉及化合物,其为(R)‑3‑(1,4‑二甲基‑1H‑苯并[d][1,2,3]三唑‑5‑基)‑3‑(3‑(((R)‑2‑乙基‑2,3‑二氢吡啶并[2,3‑f][1,4]氧氮杂环庚三烯‑4(5H)‑基)甲基)‑4‑甲基苯基)丙酸,或其药学上可接受的盐,特别是其葡甲胺盐,包含该化合物的药物组合物及其作为NRF2活化剂的用途。
USPTO Abstract
本发明涉及化合物,其为(R)‑3‑(1,4‑二甲基‑1H‑苯并[d][1,2,3]三唑‑5‑基)‑3‑(3‑(((R)‑2‑乙基‑2,3‑二氢吡啶并[2,3‑f][1,4]氧氮杂环庚三烯‑4(5H)‑基)甲基)‑4‑甲基苯基)丙酸,或其药学上可接受的盐,特别是其葡甲胺盐,包含该化合物的药物组合物及其作为NRF2活化剂的用途。
Drugs covered by this patent
- Rezlidhia (OLUTASIDENIB) · Rigel Pharms
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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