CN Patent
CN110092785A — 一种丁苯那嗪的动态拆分方法
Assigned to Guangdong HEC Pharmaceutical Co Ltd · Expires 2019-08-06 · 7y expired
What this patent protects
本发明提供一种丁苯那嗪的动态拆分方法,属于医药化工领域;所述方法可用于拆分丁苯那嗪得到(3R,11bR)‑丁苯那嗪,所述方法的特征是采用拆分试剂与丁苯那嗪混合反应,得到所需构型,分离再经过碱游离得到(3R,11bR)‑丁苯那嗪。本发明提供的分析方法能够有效分离丁苯那嗪,具有产物纯度高,收率高,操作简单,溶剂可回收等优点。
USPTO Abstract
本发明提供一种丁苯那嗪的动态拆分方法,属于医药化工领域;所述方法可用于拆分丁苯那嗪得到(3R,11bR)‑丁苯那嗪,所述方法的特征是采用拆分试剂与丁苯那嗪混合反应,得到所需构型,分离再经过碱游离得到(3R,11bR)‑丁苯那嗪。本发明提供的分析方法能够有效分离丁苯那嗪,具有产物纯度高,收率高,操作简单,溶剂可回收等优点。
Drugs covered by this patent
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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