CN Patent
CN109661393A — 帕布昔利布的新晶型及其制备方法及其用途
Assigned to Shanghai Begreat Pharmatech · Expires 2019-04-19 · 7y expired
What this patent protects
本发明公开了6‑乙酰基‑8‑环戊基‑5‑甲基‑2‑(5‑哌嗪‑1‑基‑吡啶‑2‑基氨基)‑8H‑吡啶并[2,3‑d]嘧啶‑7‑酮的新多晶型I、II、III、IV、V、VI、VII、VIII、IX、X、XI、XII和XIV及其制备方法和药用用途。晶型VIII为半水合物晶型,与现有晶型相比,新晶型在溶解度、稳定性和制备工艺方面具有明显优势。
USPTO Abstract
本发明公开了6‑乙酰基‑8‑环戊基‑5‑甲基‑2‑(5‑哌嗪‑1‑基‑吡啶‑2‑基氨基)‑8H‑吡啶并[2,3‑d]嘧啶‑7‑酮的新多晶型I、II、III、IV、V、VI、VII、VIII、IX、X、XI、XII和XIV及其制备方法和药用用途。晶型VIII为半水合物晶型,与现有晶型相比,新晶型在溶解度、稳定性和制备工艺方面具有明显优势。
Drugs covered by this patent
- Palbociclib (palbociclib) · Pfizer Inc.
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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