CN Patent

CN109593065A — 一类hdac/alk双靶点抑制剂及其制备方法与应用

Assigned to Chongqing Medical University · Expires 2019-04-09 · 7y expired

What this patent protects

本发明属于药物化学领域,具体涉及一类HDAC/ALK双靶点抑制剂及其制备方法与应用,所述HDAC/ALK双靶点抑制剂结构如式I所示,所述HDAC/ALK双靶点抑制剂对HDAC和ALK激酶具有良好的抑制活性,对HepG2肝癌细胞的抑制活性强于与目前常规的抗肝癌药物索拉菲尼相当,处于微摩尔级别。

USPTO Abstract

本发明属于药物化学领域,具体涉及一类HDAC/ALK双靶点抑制剂及其制备方法与应用,所述HDAC/ALK双靶点抑制剂结构如式I所示,所述HDAC/ALK双靶点抑制剂对HDAC和ALK激酶具有良好的抑制活性,对HepG2肝癌细胞的抑制活性强于与目前常规的抗肝癌药物索拉菲尼相当,处于微摩尔级别。

Drugs covered by this patent

Patent Metadata

Patent number
CN109593065A
Jurisdiction
CN
Classification
Expires
2019-04-09
Drug substance claim
No
Drug product claim
No
Assignee
Chongqing Medical University
Source
FDA Orange Book + USPTO grounding via Google Patents

Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.

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