CN Patent
CN109593065A — 一类hdac/alk双靶点抑制剂及其制备方法与应用
Assigned to Chongqing Medical University · Expires 2019-04-09 · 7y expired
What this patent protects
本发明属于药物化学领域,具体涉及一类HDAC/ALK双靶点抑制剂及其制备方法与应用,所述HDAC/ALK双靶点抑制剂结构如式I所示,所述HDAC/ALK双靶点抑制剂对HDAC和ALK激酶具有良好的抑制活性,对HepG2肝癌细胞的抑制活性强于与目前常规的抗肝癌药物索拉菲尼相当,处于微摩尔级别。
USPTO Abstract
本发明属于药物化学领域,具体涉及一类HDAC/ALK双靶点抑制剂及其制备方法与应用,所述HDAC/ALK双靶点抑制剂结构如式I所示,所述HDAC/ALK双靶点抑制剂对HDAC和ALK激酶具有良好的抑制活性,对HepG2肝癌细胞的抑制活性强于与目前常规的抗肝癌药物索拉菲尼相当,处于微摩尔级别。
Drugs covered by this patent
- Zykadia (ceritinib) · Novartis
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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