CN Patent
CN109516999B — 用作蛋白质激酶调节剂的化合物及其应用
Assigned to Zhejiang Taaji Hongnuo Pharmaceutical Co., Ltd. · Expires 2021-08-17 · 5y expired
What this patent protects
本发明公开了一种式Ⅰ所示的化合物,其中的各符号如权利要求中所定义。本发明的式Ⅰ所示化合物对ALK、ROS1和/或TRK激酶具有良好的抑制活性,可用于制备抑制ALK、ROS1和/或TRK激酶的药物,用于治疗癌症、疼痛、神经疾病、自身免疫疾病或发炎。
USPTO Abstract
本发明公开了一种式Ⅰ所示的化合物,其中的各符号如权利要求中所定义。本发明的式Ⅰ所示化合物对ALK、ROS1和/或TRK激酶具有良好的抑制活性,可用于制备抑制ALK、ROS1和/或TRK激酶的药物,用于治疗癌症、疼痛、神经疾病、自身免疫疾病或发炎。
Drugs covered by this patent
- Augtyro (REPOTRECTINIB) · Bristol
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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