CN Patent

CN109381440A — 一种艾乐替尼组合物

Assigned to Weihai Guanbiao Information Technology Co Ltd · Expires 2019-02-26 · 7y expired

What this patent protects

本发明涉及一种艾乐替尼口服药物,属于药物制剂技术领域。本发明所述艾乐替尼组合物,每千个单位剂量中,含有D 90 为36‑55微米的艾乐替尼150g,吐温80 4‑8g,气相二氧化硅8‑26g,硫酸钙2‑8g,羟丙基纤维素18‑32g,无水乳糖20‑46g,乙二胺四乙酸二钠4‑8g,硬脂酸镁1.0‑1.5g。本发明技术方案通过几种组分的合理配伍,一是提高了主药的溶出,二是气相二氧化硅、硫酸钙、乙二胺四乙酸二钠的联和作用,提高了储存过程中的抗吸湿性能。

USPTO Abstract

本发明涉及一种艾乐替尼口服药物,属于药物制剂技术领域。本发明所述艾乐替尼组合物,每千个单位剂量中,含有D 90 为36‑55微米的艾乐替尼150g,吐温80 4‑8g,气相二氧化硅8‑26g,硫酸钙2‑8g,羟丙基纤维素18‑32g,无水乳糖20‑46g,乙二胺四乙酸二钠4‑8g,硬脂酸镁1.0‑1.5g。本发明技术方案通过几种组分的合理配伍,一是提高了主药的溶出,二是气相二氧化硅、硫酸钙、乙二胺四乙酸二钠的联和作用,提高了储存过程中的抗吸湿性能。

Drugs covered by this patent

Patent Metadata

Patent number
CN109381440A
Jurisdiction
CN
Classification
Expires
2019-02-26
Drug substance claim
No
Drug product claim
No
Assignee
Weihai Guanbiao Information Technology Co Ltd
Source
FDA Orange Book + USPTO grounding via Google Patents

Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.

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