CN108794530A — 一种替诺福韦丙酚酰胺盐晶型及其制备方法和用途
Assigned to Shanghai Institute of Pharmaceutical Industry · Expires 2018-11-13 · 8y expired
What this patent protects
本发明公开了一种替诺福韦丙酚酰胺盐晶型及其制备方法和用途。本发明提供了一种如式I所示的替诺福韦丙酚酰胺盐的晶型甲,其X‑射线粉末衍射图在2θ值5.17±0.2°、7.30±0.2°、10.30±0.2°、10.91±0.2°、11.13±0.2°、18.55±0.2°、19.42±0.2°、21.14±0.2°和26.50±0.2°处有特征峰。该晶型具有制备简便、去除非对映异构体杂质能力强和稳定性高的优点。
USPTO Abstract
本发明公开了一种替诺福韦丙酚酰胺盐晶型及其制备方法和用途。本发明提供了一种如式I所示的替诺福韦丙酚酰胺盐的晶型甲,其X‑射线粉末衍射图在2θ值5.17±0.2°、7.30±0.2°、10.30±0.2°、10.91±0.2°、11.13±0.2°、18.55±0.2°、19.42±0.2°、21.14±0.2°和26.50±0.2°处有特征峰。该晶型具有制备简便、去除非对映异构体杂质能力强和稳定性高的优点。
Drugs covered by this patent
- Emtriva (EMTRICITABINE) · Gilead Sciences
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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