CN Patent

CN108794411B — 某些化学实体、组合物及方法

Assigned to Neupharma Inc · Expires 2022-06-07 · 4y expired

What this patent protects

本文描述了作为激酶抑制剂的基于喹喔啉的化学实体。具体而言,描述了抑制Braf突变激酶活性的含有二芳基酰胺或二芳基脲亚结构的式I的喹喔啉衍生物、含有该抑制剂化合物的药物组合物以及癌症的治疗方法,该方法包括施用有效量的Braf抑制剂化合物。

USPTO Abstract

本文描述了作为激酶抑制剂的基于喹喔啉的化学实体。具体而言,描述了抑制Braf突变激酶活性的含有二芳基酰胺或二芳基脲亚结构的式I的喹喔啉衍生物、含有该抑制剂化合物的药物组合物以及癌症的治疗方法,该方法包括施用有效量的Braf抑制剂化合物。

Drugs covered by this patent

Patent Metadata

Patent number
CN108794411B
Jurisdiction
CN
Classification
Expires
2022-06-07
Drug substance claim
No
Drug product claim
No
Assignee
Neupharma Inc
Source
FDA Orange Book + USPTO grounding via Google Patents

Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.

Track this patent

Get a daily-checked alert when vulnerability score, expiry, classification, or assignee changes. Email, Slack, or Teams delivery. Pro: 50 watches, Free: 3.