CN Patent
CN108239055B — 一种thr1442 l-天冬氨酸共晶、其制备方法及药物组合物
Assigned to Hangzhou Lingye Pharmaceutical Technology Co ltd · Expires 2023-07-18 · 3y expired
What this patent protects
本发明涉及SGLT2抑制剂THR1442(Bexagliflozin)和L‑天冬氨酸的共晶,与已知的THR1442二脯氨酸共晶相比,本发明的THR1442L‑天冬氨酸共晶具有一种或多种改进的特性。本发明还涉及THR1442L‑天冬氨酸共晶的制备方法、其药物组合物及其用于治疗受SGLT或SGLT2抑制之影响的疾病或病症的方法。
USPTO Abstract
本发明涉及SGLT2抑制剂THR1442(Bexagliflozin)和L‑天冬氨酸的共晶,与已知的THR1442二脯氨酸共晶相比,本发明的THR1442L‑天冬氨酸共晶具有一种或多种改进的特性。本发明还涉及THR1442L‑天冬氨酸共晶的制备方法、其药物组合物及其用于治疗受SGLT或SGLT2抑制之影响的疾病或病症的方法。
Drugs covered by this patent
- Brenzavvy (BEXAGLIFLOZIN) · Theracosbio
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
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