CN Patent
CN108129514A — 磷酸/膦酸衍生物的单一异构体及其医药用途
Assigned to BEIJING MEIBEITA PHARMACEUTICAL RESEARCH Co Ltd · Expires 2018-06-08 · 8y expired
What this patent protects
本发明涉及式Ia所示的磷酸/膦酸衍生物及其非毒性药学上可接受的盐;其中,式Ib所示的非对映异构体的含量小于2%: 结构式Ia和Ib中,Ar代表取代或未取代的苯环或萘环,R 1 代表H或碳原子数1‑6的烷基;R 2 代表碳原子数1‑6的烷基或环烷基;D代表含磷酸/膦酸基的药理活性分子的残基,即 代表含磷酸/膦酸基的药理活性分子。
USPTO Abstract
本发明涉及式Ia所示的磷酸/膦酸衍生物及其非毒性药学上可接受的盐;其中,式Ib所示的非对映异构体的含量小于2%: 结构式Ia和Ib中,Ar代表取代或未取代的苯环或萘环,R 1 代表H或碳原子数1‑6的烷基;R 2 代表碳原子数1‑6的烷基或环烷基;D代表含磷酸/膦酸基的药理活性分子的残基,即 代表含磷酸/膦酸基的药理活性分子。
Drugs covered by this patent
- Emtriva (EMTRICITABINE) · Gilead Sciences
Bibliographic data sourced from FDA Orange Book + USPTO public records. Plain-English summary generated by AI grounded in source text. Patent term extensions (PTR, SPC, pediatric) may shift the effective expiry. Not legal advice.
Track this patent
Get a daily-checked alert when vulnerability score, expiry, classification, or assignee changes. Email, Slack, or Teams delivery. Pro: 50 watches, Free: 3.